GSK3368715 (dihydrochloride), CAS [[1628925-77-8]]
Catalog Number:
MCE-HY-128717A
| Article Name: |
GSK3368715 (dihydrochloride), CAS [[1628925-77-8]] |
| Biozol Catalog Number: |
MCE-HY-128717A |
| Supplier Catalog Number: |
HY-128717A |
| Alternative Catalog Number: |
MCE-HY-128717A-10MMX1ML,MCE-HY-128717A-25MG,MCE-HY-128717A-50MG,MCE-HY-128717A-10MG,MCE-HY-128717A-1MG,MCE-HY-128717A-5MG,MCE-HY-128717A-100MG |
| Manufacturer: |
MedchemExpress |
| Category: |
Biochemikalien |
| Alternative Names: |
EPZ019997 (dihydrochloride) |
| GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)). GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) produces a shift in arginine methylation states, alters exon usage, and has strong anti-cancer activity[1]. |
| Molecular Weight: |
439.46 |
| Purity: |
99.96 |
| CAS Number: |
[1628925-77-8] |
| Formula: |
C20H40Cl2N4O2 |
| Target: |
Histone Methyltransferase |
| Application Notes: |
MCE Product type: Reference compound |
