GSK3368715 (hydrochloride), CAS [[2227587-25-7]] Preis auf Anfrage

Product Overview

• Article Name: GSK3368715 (hydrochloride), CAS [[2227587-25-7]] Preis auf Anfrage
• Biozol Catalog Number: MCE-HY-128717C
• Supplier Catalog Number: HY-128717C
• Alternative Catalog Number: MCE-HY-128717C-1UNIT
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: EPZ019997 (hydrochloride)

Product Description

GSK3368715 (EPZ019997) hydrochloride is an orally active, reversible, SAM-noncompetitive type I protein arginine methyltransferase (PRMT) inhibitor with IC50 values of 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), and 1.7 nM (PRMT8). GSK3368715 hydrochloride induces a shift in arginine methylation states, alters exon usage, and exhibits potent anticancer activity[1].

Product Properties

• Molecular Weight: 403.00
• CAS Number: [2227587-25-7]
• Formula: C20H39ClN4O2
• Target: Histone Methyltransferase

Application Notes

• Application Notes: MCE Product type: Reference compound