PF 05089771 tosylate is a potent, orally active and selective arylsulfonamide Nav1.7 inhibitor, with IC50 values of 11 nM, 12 nM, 13 nM, 171 nM and 8 nM for hNav1.7, cynNav1.7, dogNav1.7, ratNav1.7, and musNav1.7, respectively. PF 05089771 is under the study for pain and diabetic neuropathy[1][2].
Molecular Weight:
672.56
CAS Number:
[1430806-04-4]
Formula:
C25H20Cl2FN5O6S3
Target:
Sodium Channel
Application Notes:
MCE Product type: Reference compound
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