(E/Z)-CLH304a (GABAB receptor antagonist 1) is a mixture of (E)-CLH304a and (Z)-CLH304a. (E)-CLH304a (CLH304a, HY-129636) is a specific and noncompetitive GABAB receptor negative allosteric modulator (NAM). CLH304a inhibits Baclofen (HY-B0007)-induced ERK1/2 phosphorylation in HEK293 cells overexpressing GABAB receptors[1][2].
Molecular Weight:
304.38
CAS Number:
[797-17-1]
Formula:
C18H24O4
Target:
ERK,GABA Receptor
Application Notes:
MCE Product type: Reference compound
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