VPC12249 is a competitive dual LPA1/LPA3 antagonist with Ki values of 137nM and 428 nM, respectively. VPC12249 inhibits calcium mobilization in HEK293T cells with a Ki value of ~130 nM. VPC12249 is promising for research of ovarian cancer and hypertensive diseases[1].
Molecular Weight:
601.75
CAS Number:
[403520-23-0]
Formula:
C34H52NO6P
Target:
LPL Receptor
Application Notes:
MCE Product type: Reference compound
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