JHU37160, CAS [[2369979-68-8]]

Catalog Number: MCE-HY-131881
Article Name: JHU37160, CAS [[2369979-68-8]]
Biozol Catalog Number: MCE-HY-131881
Supplier Catalog Number: HY-131881
Alternative Catalog Number: MCE-HY-131881-5MG,MCE-HY-131881-25MG,MCE-HY-131881-10MMX1ML,MCE-HY-131881-100MG,MCE-HY-131881-10MG,MCE-HY-131881-50MG
Manufacturer: MedchemExpress
Category: Biochemikalien
JHU37160 is a potent and brain-penetrant DREADD agonist, with EC50s of 18.5 nM and 0.2 nM for hM3Dq and hM4Di DREADDs in HEK-293 cells, respectively. JHU37160 exhibits selective [3H]Clozapine displacement from DREADDs and not from other Clozapine-binding sites in mice brain tissue[1].
Molecular Weight: 358.84
Purity: 99.98
CAS Number: [2369979-68-8]
Formula: C19H20ClFN4
Target: mAChR
Application Notes: Reference compound