EST64454 maleate is a highly soluble sigma1 receptor antagonist, demonstrating potent antinociceptive properties for pain treatment. EST64454 maleate exhibits excellent metabolic stability across various species and possesses an adequate pharmacokinetic profile in rodents. EST64454 maleate has been identified as a promising clinical candidate due to its favorable aqueous solubility and high permeability in Caco-2 cells.
Molecular Weight:
480.46
CAS Number:
[2088272-67-5]
Formula:
C22H26F2N4O6
Target:
Sigma Receptor
Application Notes:
MCE Product type: Reference compound
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