DYRK1-IN-1 is a highly selective and ligand-efficient DYRK1A inhibitor. DYRK1-IN-1 inhibits DYRK1A phosphorylation activity with an IC50 value of 220 nM. DYRK1-IN-1 can be used for the research of central nervous system penetrant DYRK1A chemical probe[1].
Molecular Weight:
240.26
Purity:
99.71
CAS Number:
[2814486-79-6]
Formula:
C12H12N6
Target:
DYRK
Application Notes:
MCE Product type: Reference compound1
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