WDR5-IN-1 is a potent and selective WD repeat domain 5 (WDR5) inhibitor, with a Kd of 50 of 2.2 nM. WDR5-IN-1 diminishes MYC recruitment at WDR5-displaced genes and exhibits potent anti-proliferative effects in CHP-134 (neuroblastoma) and Ramos (Burkitts lymphoma) lines[1].
Molecular Weight:
514.59
Purity:
98
CAS Number:
[2408842-51-1]
Formula:
C30H31FN4O3
Target:
Apoptosis,WDR5
Application Notes:
MCE Product type: Reference compound
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