PKCbeta inhibitor 1 is a potent, ATP-competitive, and selective PKCbeta inhibitor with IC50s of 21 and 5 nM for human PKCbeta1 and PKCbeta2, respectively. PKCbeta inhibitor 1 exhibits selectivity of more than 60-fold in favor of PKCbeta2 relative to other PKC isozymes (PKCalpha, PKCgamma, and PKCepsilon)[1][2].
Molecular Weight:
411.46
Purity:
99.40
CAS Number:
[257879-35-9]
Formula:
C24H21N5O2
Target:
Apoptosis,PKC
Application Notes:
MCE Product type: Reference compound
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