EST73502 is a selective, orally active and blood-brain barrier (BBB) penetrant dual µ-opioid receptor (MOR) agonist and sigma1 receptor (sigma1R) antagonist, with Kis of 64 nM and 118 nM for MOR and sigma1R, respectively. EST73502 has antinociceptive activity[1].
Molecular Weight:
352.42
CAS Number:
[1838622-25-5]
Formula:
C19H26F2N2O2
Target:
Opioid Receptor,Sigma Receptor
Application Notes:
MCE Product type: Reference compound
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