NAS-181 (free base), CAS [[205242-61-1]] Preis auf Anfrage

Product Overview

• Article Name: NAS-181 (free base), CAS [[205242-61-1]] Preis auf Anfrage
• Biozol Catalog Number: MCE-HY-135507A
• Supplier Catalog Number: HY-135507A
• Alternative Catalog Number: MCE-HY-135507A-1UNIT
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

NAS181 free base is a potent and selective antagonist of rat 5-HT1B receptor, with a Ki of 47 nM. NAS181 free base shows 13-fold selectivity for r5-HT1B over bovine 5-HT1B receptor (Ki=630 nM). NAS181 free base increases the 5-HT turnover and the synaptic concentration of 5-HT by inhibiting terminal r5-HT1B autoreceptors[1][2].

Product Properties

• Molecular Weight: 346.42
• CAS Number: [205242-61-1]
• Formula: C19H26N2O4
• Target: 5-HT Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound