TAN-452, CAS [[892039-23-5]]

Product Overview

• Article Name: TAN-452, CAS [[892039-23-5]]
• Biozol Catalog Number: MCE-HY-136208
• Supplier Catalog Number: HY-136208
• Alternative Catalog Number: MCE-HY-136208-100MG,MCE-HY-136208-50MG,MCE-HY-136208-10MG,MCE-HY-136208-10MMX1ML,MCE-HY-136208-25MG,MCE-HY-136208-5MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

TAN-452 is an orally active, selective peripherally acting delta-opioid receptor (DOR) antagonist with a Ki of 0.47 nM and a Kb of 0.21 nM. TAN-452 is an antagonist for µ-opioid receptor (MOR, Ki=36.56 nM and Kb=9.43 nM) and kappa-opioid receptor (KOR, Ki=5.31 nM and Kb=7.18 nM). TAN-452, a derivative of Naltrindole, demonstrates low brain penetrability and attenuates morphine-induced side effects without affecting pain control[1].

Product Properties

• Molecular Weight: 486.56
• Purity: 99.44
• CAS Number: [892039-23-5]
• Formula: C29H30N2O5
• Target: Opioid Receptor

Application Notes

• Application Notes: Reference compound