PHD-1-IN-1 is an orally active and potent HIF prolylhydroxylase domain-1 (PHD-1) inhibitor with an IC50 of 0.034 µM. PHD-1-IN-1 has a unique monodentate binding interaction with the active site Fe2+ ion and induces the formation of an Arg367-out pocket[1].
Molecular Weight:
220.23
Purity:
99.54
CAS Number:
[2009343-14-8]
Formula:
C13H8N4
Target:
HIF/HIF Prolyl-Hydroxylase
Application Notes:
Reference compound
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