GLS1 Inhibitor-1 (Compound 27) is an orally active inhibitor for glutaminase 1 (GLS1) with an IC50 of 0.021 µM. GLS1 Inhibitor-1 inhibits the proliferation of PC-3 with an IC50 of 0.3 nM. GLS1 Inhibitor-1 exhibits antitumor efficacy against NCI-H1703 with GI50 of 0.011 µM. GLS1 Inhibitor-1 exhibits moderate pharmacokinetic characteristics[1].
Molecular Weight:
411.48
Purity:
98.5
CAS Number:
[1832646-52-2]
Formula:
C19H21N7O2S
Target:
Glutaminase
Application Notes:
MCE Product type: Reference compound1
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