GSK620, a chemical probe, is a potent and orally active pan-BD2 inhibitor with excellent broad selectivity, developability and in vivo oral pharmacokinetics. GSK620 is highly selective for the BET-BD2 family of proteins, with >200-fold selectivity over all other bromodomains. GSK620 shows an anti-inflammatory phenotype in human whole blood[1].
Molecular Weight:
325.36
Purity:
99.79
CAS Number:
[2088410-46-0]
Formula:
C18H19N3O3
Target:
Epigenetic Reader Domain
Application Notes:
MCE Product type: Reference compound
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