(R)-PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC50 value of 1.8 µM. (R)-PS210 targets to the PIF-binding pocket of PDK1. PIF: The protein kinase C-related kinase 2 (PRK2)-interacting fragment[1].
Molecular Weight:
380.31
Purity:
98.09
CAS Number:
[1410101-89-1]
Formula:
C19H15F3O5
Target:
PDK-1
Application Notes:
MCE Product type: Reference compound
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