EZH2-IN-4 is an orally active, potent EZH2 inhibitor with IC50s of 0.923 nM and 2.65 nM against wild type (WT) 5-membered (5-mer) EZH2 and mutant 5-mer EZH2, respectively. EZH2-IN-4 has anti-cancer activity[1].
Molecular Weight:
511.72
CAS Number:
[2088132-99-2]
Formula:
C29H41N3O3S
Target:
Histone Methyltransferase
Application Notes:
MCE Product type: Reference compound
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