Sulfopin (PIN1-3) is a highly selective covalent inhibitor of Pin1 with an apparent Ki of 17 nM. Sulfopin blocks Myc-driven tumors in vivo. The peptidyl-prolyl isomerase, Pin1, is exploited in cancer to activate oncogenes and inactivate tumor suppressors[1].
Molecular Weight:
281.81
Purity:
99.82
CAS Number:
[2451481-08-4]
Formula:
C11H20ClNO3S
Target:
PIN1
Application Notes:
MCE Product type: Reference compound
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