Siramesine (fumarate), CAS [[163630-79-3]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-14221B
Supplier Catalog Number:
HY-14221B
Alternative Catalog Number:
MCE-HY-14221B-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Alternative Names:
LU-28-179 (fumarate)
Siramesine (Lu 28-179) fumarate is a potent sigma-2 receptor agonist. Siramesine fumarate has a subnanomolar affinity for sigma-2 receptors (IC50=0.12 nM) and exhibits a 140-fold selectivity for sigma-2 receptors over sigma-1 receptors (IC50=17 nM). Siramesine fumarate triggers cell death through destabilisation of mitochondria, but not lysosomes. Anti-cancer activity[1][2][3].
Molecular Weight:
570.65
CAS Number:
[163630-79-3]
Formula:
C34H35FN2O5
Target:
Sigma Receptor
Application Notes:
MCE Product type: Reference compound
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