SB 271046 (Hydrochloride) (Standard) is the analytical standard of SB 271046 (Hydrochloride). This product is intended for research and analytical applications. SB 271046 Hydrochloride (SB 271046A) is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 9.02, 8.55, and 8.81 for rat, pig and human, respectively. SB 271046 Hydrochloride is over 200 fold selective for the 5-HT6 receptor vs 55 other receptors, binding sites and ion channels. Anticonvulsant activity (EC50=0.16 µM)[1].
Molecular Weight:
488.45
CAS Number:
[209481-24-3]
Formula:
C20H23Cl2N3O3S2
Target:
5-HT Receptor,Reference Standards
Application Notes:
MCE Product type: Reference Standards
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