CM398 is a highly selective, orally active sigma-2 receptor ligand (Ki=0.43 nM), with high sigma-1/sigma-2 selectivity rato (1000-fold). CM398 shows notable affinity for dopamine (Ki=32.90 nM) and serotonin transporters (Ki=244.2 nM). CM398 shows promising anti-inflammatory analgesic effects in the formalin model of inflammatory pain in mice[1].
Molecular Weight:
395.49
Purity:
99.85
CAS Number:
[1121931-70-1]
Formula:
C23H29N3O3
Target:
Sigma Receptor
Application Notes:
Reference compound
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