PERK-IN-5 is a highly potent, selectively and orally bioavailable PERK inhibitor (IC50s of 2 and 9 nM for PERK and p-eIF2alpha, respectively). PERK-IN-5 can significantly inhibit tumor growth in the 786-O renal cell carcinoma xenograft tumor model[1].
Molecular Weight:
468.50
Purity:
99.40
CAS Number:
[2616821-91-9]
Formula:
C25H26F2N4O3
Target:
PERK
Application Notes:
MCE Product type: Reference compound
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