S1427 is a tranylcypromine-derived LSD1 inhibitor with the IC50 of 390 nM and Ki of 80 nM. S1427 exhibits desirable hERG channel inhibition and microsomal stability profiles. Inhibition of LSD1 partially reduces the proliferation of cancer cells[1].
Molecular Weight:
474.52
CAS Number:
[2447061-40-5]
Formula:
C25H29F3N4O2
Target:
Histone Demethylase
Application Notes:
MCE Product type: Reference compound
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