Androgen receptor antagonist 5, CAS [[2586195-28-8]] Preis auf Anfrage

Catalog Number: MCE-HY-146494
Article Name: Androgen receptor antagonist 5, CAS [[2586195-28-8]] Preis auf Anfrage
Biozol Catalog Number: MCE-HY-146494
Supplier Catalog Number: HY-146494
Alternative Catalog Number: MCE-HY-146494-1UNIT
Manufacturer: MedchemExpress
Category: Biochemikalien
Androgen receptor antagonist 5 (compound 42f) is a potent androgen receptor (AR) antagonist with an IC50 value of 6.17 µM. Androgen receptor antagonist 5 can effectively impair AR nuclear translocation, reducing the levels of nuclear AR, and disrupts AR-mediated gene regulation. Androgen receptor antagonist 5 has antiproliferative activity against LNCaP and exhibits antitumor activity in LNCaP xenograft tumor mice model. Androgen receptor antagonist 5 can be used for researching prostate cancer[1].
Molecular Weight: 493.43
CAS Number: [2586195-28-8]
Formula: C21H15F4N5O3S
Target: Androgen Receptor
Application Notes: MCE Product type: Reference compound1