Lirafugratinib (hydrochloride), CAS [[2688040-45-9]]

Product Overview

• Article Name: Lirafugratinib (hydrochloride), CAS [[2688040-45-9]]
• Biozol Catalog Number: MCE-HY-147250A
• Supplier Catalog Number: HY-147250A
• Alternative Catalog Number: MCE-HY-147250A-50MG,MCE-HY-147250A-100MG,MCE-HY-147250A-10MG,MCE-HY-147250A-25MG,MCE-HY-147250A-10MMX1ML,MCE-HY-147250A-5MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: RLY-4008 (hydrochloride)

Product Description

Lirafugratinib (RLY-4008) hydrochloride is an orally active, irreversible and highly selective FGFR2 inhibitor with an IC50 of 3 nM. Lirafugratinib hydrochloride covalently binds to Cys491. Lirafugratinib hydrochloride targets FGFR2 primary alterations and resistance mutations and induces tumor regression while sparing other FGFRs[1].

Product Properties

• Molecular Weight: 546.00
• Purity: 98.96
• CAS Number: [2688040-45-9]
• Formula: C28H25ClFN7O2
• Target: FGFR

Application Notes

• Application Notes: MCE Product type: Reference compound