Rolapitant (SCH619734) is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a Ki of 0.66 nM. Rolapitant does not interact with CYP3A4. Rolapitant shows potent anti-emetic activity in a ferret emesis model[1][2].
Molecular Weight:
500.48
Purity:
99.89
CAS Number:
[552292-08-7]
Formula:
C25H26F6N2O2
Target:
Neurokinin Receptor
Application Notes:
MCE Product type: Reference compound
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