MPO-IN-5 (compound 1) is a potent, irreversible MPO (myeloperoxidase) inhibitor. MPO-IN-5 inhibits MPO peroxidation and hERG binding, with IC50 values of 0.22 and 2.8 µM, respectively. MPO-IN-5 shows rapid kinetics of inhibition, with enzyme inactivation rate (kinact/Ki) of 23000 M-1s-1[1].
Molecular Weight:
428.49
CAS Number:
[2476764-11-9]
Formula:
C24H24N6O2
Target:
Glutathione Peroxidase,Potassium Channel
Application Notes:
MCE Product type: Reference compound
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