PPARgamma phosphorylation inhibitor 1, CAS [[2882975-84-8]]

Product Overview

• Article Name: PPARgamma phosphorylation inhibitor 1, CAS [[2882975-84-8]]
• Biozol Catalog Number: MCE-HY-147705
• Supplier Catalog Number: HY-147705
• Alternative Catalog Number: MCE-HY-147705-5MG,MCE-HY-147705-50MG,MCE-HY-147705-25MG,MCE-HY-147705-10MG,MCE-HY-147705-10MMX1ML,MCE-HY-147705-100MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

PPARgamma phosphorylation inhibitor 1 (Compound 10) is a potent PPARgamma binder with the IC50 of 24 nM. PPARgamma phosphorylation inhibitor 1 inhibits CDK5-mediated phosphorylation of PPARgamma Ser273 with the IC50 of 160 nM. PPARgamma phosphorylation inhibitor 1 displays negligible PPARgamma agonism in a reporter gene assay. Antidiabetic effects[1].

Product Properties

• Molecular Weight: 441.26
• Purity: 99.81
• CAS Number: [2882975-84-8]
• Formula: C22H14Cl2N2O4
• Target: PPAR

Application Notes

• Application Notes: MCE Product type: Reference compound