BMS-684 is a selective DGKalpha inhibitor with an IC50 of 15 nM. BMS-684 inhibits DGKalpha kinase activity with >100-fold selectivity over the related DGK type I family members DGKbeta and DGKgamma. BMS-684 does not inhibit any of the other seven DGK isozymes[1].
Molecular Weight:
454.52
Purity:
99.76
CAS Number:
[313552-29-3]
Formula:
C27H26N4O3
Target:
DGK
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted