A2AR-antagonist-1, CAS [[2922920-71-4]]

Product Overview

• Article Name: A2AR-antagonist-1, CAS [[2922920-71-4]]
• Biozol Catalog Number: MCE-HY-149916
• Supplier Catalog Number: HY-149916
• Alternative Catalog Number: MCE-HY-149916-100MG,MCE-HY-149916-5MG,MCE-HY-149916-10MMX1ML,MCE-HY-149916-50MG,MCE-HY-149916-10MG,MCE-HY-149916-25MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

A2AR-antagonist-1 (compound 38) is an orally active adenosine A2A receptor (A2AR) antagonist (IC50=29 nM). A2AR-antagonist-1 exhibits anti-tumor activity and mouse liver microsomal metabolic stability (t1/2=86.1 min). A2AR-antagonist-1 is also a T cells activator, via inhibiting immunosuppressive molecules (LAG-3 and TIM-3) and enhancing effector molecules (GZMB, IFNG, and IL-2)[1].

Product Properties

• Molecular Weight: 451.52
• Purity: 96.68
• CAS Number: [2922920-71-4]
• Formula: C27H25N5O2
• Target: Adenosine Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound