HDAC-IN-57 is an orally active inhibitor of histone deacetylases (HDAC), with IC50s of 2.07 nM, 4.71 nM, 2.4 nM and 107 nM for HDAC1, HDAC2, HDAC6, HDAC8, respectively. HDAC-IN-57 can inhibits LSD1, with IC50 of 1.34 µM. HDAC-IN-57 induces apoptosis, and has anti-tumor activity[1].
Molecular Weight:
377.39
CAS Number:
[2716217-79-5]
Formula:
C21H19N3O4
Target:
Apoptosis,HDAC,Histone Demethylase
Application Notes:
MCE Product type: Reference compound
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