MK-0429 (L-000845704) is an orally active, potent, selective and nonpeptide pan-integrin antagonist with IC50 values of 1.6 nM, 2.8 nM, 0.1 nM, 0.7 nM, 0.5 nM and 12.2 nM for alphavbeta1, alphavbeta3, alphavbeta5, alphavbeta6, alphavbeta8 and alpha5beta1, respectively[1][2][3].
Molecular Weight:
439.51
Purity:
99.50
CAS Number:
[227963-15-7]
Formula:
C23H29N5O4
Target:
Integrin
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted