GRP78-IN-3 (Compound 8) is a selective Grp78 (HSPA5) inhibitor with an IC50 of 0.59 µM. GRP78-IN-3 is 7-fold selective for HspA5 compared to HspA9 (IC50 of 4.3 µM) and >20-fold selective for HspA5 compared to HspA2 (IC50 of 13.9 µM)[1].
Molecular Weight:
342.42
Purity:
99.88
CAS Number:
[2707510-30-1]
Formula:
C17H18N4O2S
Target:
HSP
Application Notes:
MCE Product type: Reference compound
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