GZ-11608 is a potent and selective vesicular monoamine transporter-2 (VMAT2) inhibitor with high affinity (Ki = 25 nM). GZ-11608 decreases methamphetamine-induced dopamine release from isolated synaptic vesicles from brain dopaminergic neurons. GZ-11608 exhibits rapid brain penetration and without neurotoxicity. GZ-11608 can be used for the research of methamphetamine use disorder[1].
Molecular Weight:
283.41
CAS Number:
[2141974-01-6]
Formula:
C19H25NO
Target:
Monoamine Transporter
Application Notes:
MCE Product type: Reference compound
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