CB2R antagonist 3 is a selective antagonist of cannabinoid type 2 receptor (CB2R). CB2R antagonist 3 has high affinity for human CB2R and specific selectivity for CB1R. CB2R antagonist 3 can be combined with CB65 (HY-110047), the activator of CB2R. CB2R antagonist 3 effectively up-regulates the expression of anti-inflammatory cytokines and down-regulates the expression of pro-inflammatory cytokines[1].
Molecular Weight:
410.64
Purity:
98.08
Formula:
C27H42N2O
Target:
Cannabinoid Receptor
Application Notes:
MCE Product type: Reference compound
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