RK-701 is an highly selective and non-genotoxic inhibitor of G9a with IC50 value of 23-27 nM. RK-701 selectively up-regulates HbF, gamma- Globin, BGLT3 expression, down-regulates H3K9me2 expression. RK-701 also has inhibition for BCL11A and ZBTB7A[1].
Molecular Weight:
446.54
Purity:
98.04
CAS Number:
[2648855-18-7]
Formula:
C26H30N4O3
Target:
Histone Methyltransferase
Application Notes:
MCE Product type: Reference compound
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