Rimegepant, CAS [[1289023-67-1]]

Product Overview

• Article Name: Rimegepant, CAS [[1289023-67-1]]
• Biozol Catalog Number: MCE-HY-15498
• Supplier Catalog Number: HY-15498
• Alternative Catalog Number: MCE-HY-15498-10MMX1ML, MCE-HY-15498-5MG, MCE-HY-15498-10MG, MCE-HY-15498-25MG, MCE-HY-15498-50MG, MCE-HY-15498-100MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: BMS-927711, BHV-3000

Product Description

Rimegepant (BMS-927711) is an orally bioavailable and blood-brain barrier permeable antagonist of CGRP and AMY1 receptors, with a pIC50 of 8.01 and a Ki of 0.027 nM for human CGRP receptors. Rimegepant antagonizes cAMP production induced by alphaCGRP, betaCGRP and amylin at CGRP and AMY1 receptors in humans, rats and mice, as well as at rat AMY3 receptors. Rimegepant can be used in research related to migraine[1].

Product Properties

• Molecular Weight: 534.56
• Purity: 99.99
• CAS Number: [1289023-67-1]
• Formula: C28H28F2N6O3
• Target: CGRP Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound