CARM1 degrader-1 (hydrochloride)

Catalog Number: MCE-HY-156152A
Article Name: CARM1 degrader-1 (hydrochloride)
Biozol Catalog Number: MCE-HY-156152A
Supplier Catalog Number: HY-156152A
Alternative Catalog Number: MCE-HY-156152A-10MG,MCE-HY-156152A-25MG,MCE-HY-156152A-1MG,MCE-HY-156152A-5MG,MCE-HY-156152A-50MG,MCE-HY-156152A-100MG
Manufacturer: MedchemExpress
Category: Biochemikalien
CARM1 degrader-1 hydrochloride is a CARM1 PROTAC degrader (DC50 = 8.1 nM) with high selectivity over other protein arginine methyltransferases. CARM1 degrader-1 hydrochloride degrades CARM1 in a VHL- and proteasome-dependent manner. CARM1 degrader-1 hydrochloride downregulates the methylation level of CARM1 substrates in cell-based assays. CARM1 degrader-1 hydrochloride inhibits cancer cell migration in cell-based assays. CARM1 degrader-1 hydrochloride can be used in breast cancer research[1].
Molecular Weight: 1316.14
Purity: 99.44
Formula: C71H99ClN12O8S
Target: Histone Methyltransferase,PROTACs
Application Notes: MCE Product type: Reference compound