GSK2801, a chemical probe, is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with Kd values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4[1].
Molecular Weight:
371.45
Purity:
99.95
CAS Number:
[1619994-68-1]
Formula:
C20H21NO4S
Target:
Apoptosis,Epigenetic Reader Domain
Application Notes:
MCE Product type: Reference compound1
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