TPT-004 is a selective and oraly active tryptophan hydroxylases (TPH) inhibitor with IC50s of 77 nM and 16 nM for TPH1 and TPH2, repsectively. TPT-004 exhibits exceptional selectivity for TPH1 compared with other members of the AAAH family. TPT-004 shows efficacy peripheral serotonin attenuation and colorectal tumor growth in mice[1][2].
Molecular Weight:
400.45
Purity:
99.90
CAS Number:
[3032648-15-7]
Formula:
C18H20N6O3S
Target:
Tryptophan Hydroxylase
Application Notes:
MCE Product type: Reference compound
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