Brexpiprazole-d8-1, CAS [[1427049-19-1]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-15780S1
Supplier Catalog Number:
HY-15780S1
Alternative Catalog Number:
MCE-HY-15780S1-500UG,MCE-HY-15780S1-1MG
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Alternative Names:
OPC-34712-d8-1
Brexpiprazole-d8-1 (OPC-34712-d8-1) is the deuterium labeled Brexpiprazole (HY-15780)[1]. Brexpiprazole (OPC-34712), an atypical orally active antipsychotic agent, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic alpha1B (Ki=0.17 nM) and alpha2C receptors (Ki=0.59 nM)[2][3].
