BQ-788 is a potent, selective ETB receptor antagonist with IC50 of 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells, poorly inhibiting the binding to ETA receptors in human neuroblastoma cell line SK-N-MC cells with IC50 of 1300 nM[1].
Molecular Weight:
641.80
Purity:
99.70
CAS Number:
[173326-37-9]
Formula:
C34H51N5O7
Target:
Endothelin Receptor
Application Notes:
Reference compound
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