Aprocitentan, CAS [[1103522-45-7]]

Product Overview

• Article Name: Aprocitentan, CAS [[1103522-45-7]]
• Biozol Catalog Number: MCE-HY-15895
• Supplier Catalog Number: HY-15895
• Alternative Catalog Number: MCE-HY-15895-5MG,MCE-HY-15895-1MG,MCE-HY-15895-25MG,MCE-HY-15895-10MMX1ML,MCE-HY-15895-50MG,MCE-HY-15895-100MG,MCE-HY-15895-10MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: ACT-132577

Product Description

Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is an orally active dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively. Aprocitentan is an antihypertensive agent[1].

Product Properties

• Molecular Weight: 546.19
• Purity: 99.55
• CAS Number: [1103522-45-7]
• Formula: C16H14Br2N6O4S
• Target: Endothelin Receptor

Application Notes

• Application Notes: Reference compound