Aprocitentan-d4 is a deuterium labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is an orally active dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively. Aprocitentan is an antihypertensive agent[1].
Molecular Weight:
550.22
Purity:
97.39
Formula:
C16H10D4Br2N6O4S
Target:
Endothelin Receptor,Isotope-Labeled Compounds
Application Notes:
Isotope-Labeled Compounds
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