RN-1665 is an orally active TRPV4 antagonist that exhibits excellent selectivity for related TRP receptors such as TRPV1, TRPV3 and TRPM8. RN-1665 is a TRPV4 probe for focus screens, with IC50s of 0.26 µM and 0.39 µM for hTRPV4 and rTRPV4 from human and rat, respectively[1].
Molecular Weight:
513.54
Purity:
99.93
CAS Number:
[1803003-65-7]
Formula:
C20H24F5N3O3S2
Target:
TRP Channel
Application Notes:
MCE Product type: Reference compound
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