uPSEM792 is a pharmacologically selective effector molecules (PSEM) agonist for PSAM4-GlyR, with an affinity of Ki of 0.7 nM. uPSEM792 is a substrate for efflux transporters in brains of wild type and dual P-gp and BCRP knockout mice. uPSEM7952 is a possible lead for developing the PET radioligand for PSAM4-GlyR[1].
Molecular Weight:
241.29
Purity:
99.92
CAS Number:
[2323525-19-3]
Formula:
C14H15N3O
Target:
5-HT Receptor
Application Notes:
Reference compound
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