TRPV1 antagonist 6 (compound 51) is a mode-selective antagonist for transient receptor potential vanilloid member 1 (TRPV1), which shows antagonism with IC50 of 2.85 nM to capsaicin activation and 28.48 % inhibition against proton activation at a 3 µM concentration[1].
Molecular Weight:
493.99
Formula:
C26H28ClN5O3
Target:
TRP Channel
Application Notes:
Reference compound
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