GS-9770 is an orally active inhibitor for HIV protease with Ki of 0.16 nM. GS-9770 exhibits antiviral activity aginst HIV-1 strains and HIV-2 strains with EC50 of 1.9-26 nM, and 26 nM. GS-9770 is metabolic stable in human liver microsomes. GS-9770 exhibits good pharmacokinetic characters in Sprague Dawley rats[1].
Molecular Weight:
811.15
CAS Number:
[2306328-43-6]
Formula:
C35H34ClF7N10O3
Target:
HIV Protease
Application Notes:
MCE Product type: Reference compound
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