alpha2A-AR agonist 1 (Compound B9) is a selective agonist for alpha2-adrenergic receptor (alpha2A-AR) with EC50 of 0.23 nM. alpha2A-AR agonist 1 exhibits a hypnotic effect, with ED50 of 0.138 mg/kg in the loss of righting reflex (LORR) experiment. alpha2A-AR agonist 1 exhibits metabolic stability in mouse liver microsomes[1].
Molecular Weight:
279.13
Purity:
99.92
CAS Number:
[2971825-58-6]
Formula:
C12H11BrN2O
Target:
Adrenergic Receptor
Application Notes:
MCE Product type: Reference compound
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